Bioactive Small Molecules

A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.

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6,241 – 6,255 of 60,541 results

6,241

Medchemexpress LLC Spiroxamine | 118134-30-8 | 99.9% | 50 MG

Spiroxamine analytical standard (CAS 118134-30-8) is supplied as a high-purity liquid reference material for analytical and residue testing. It is intended for method development, calibration, and quantitative analyses using HPLC, GC, and MS.

High purity of 99.9% (COA available).
Suitable as an analytical reference for HPLC, GC, and MS.
Molecular formula C18H35NO2; molecular weight 297.48 g/mol.
Available in small pack sizes suitable for analytical workflows.
SDS and certificate of analysis available for quality verification.

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6,242

Medchemexpress LLC Fluralaner (Standard) | 864731-61-3 | 100.0% | 556.29 | 25 MG

Fluralaner (Standard) is the analytical standard of Fluralaner. It is intended for research and analytical applications. Fluralaner (INN) is a systemic insecticide and acaricide that works through potent blockage of GABA and L-glutamate gated chloride channels. It is for research use only and not sold to patients.

Serves as a reference standard for assays
Commonly used in qualitative, quantitative, and methodological research experiments such as HPLC, GC, and MS

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6,243

Cayman Chemical Camellianin A, Purity: ≥95%, CAS: 109232-77-1, 5 mg

A flavonoid with diverse biological activities; inhibits ACE by 30.16% at 500 µg/ml; induces cell cycle arrest at the G1 phase and apoptosis in HepG2 and MCF-7 cells at 200 µM; reduces hepatocyte apoptosis, as well as hepatic TNF-α, IL-6, IL-1β, and MDA levels, in a mouse model of carbon tetrachloride-induced liver injury at 30 mg/kg

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6,244

Cayman Chemical Poloxin, Purity: ≥98%, CAS: 321688-88-4, 50 mg

An inhibitor of the Plk1 polo-box domain (apparent IC50 = 4.8 µM); selective for the Plk1 PBD over Plk2 and Plk3 PBDs (IC50s = 18.7 and 53.9 µM, respectively); induces cell cycle arrest at the G2/M phase, apoptosis, and mislocalization of Plk1 in HeLa cells at 5, 10, and 25 µM; reduces cell proliferation in a panel of 10 cancer cell lines (EC50s = 15-35 µM); reduces tumor growth and induces intratumor apoptosis in an MDA-MB-231 mouse xenograft model at 40 mg/kg

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6,245

Cayman Chemical Neoeriocitrin, Purity: ≥98%, CAS: 888471-94-1, 5 mg

A flavonoid; inhibits the production of DPPH radicals by 17.2% and the formation of superoxide radicals by 48.3% in cell-free assays; decreases the rate of LDL oxidation ex vivo in isolated hamster plasma; increases proliferation of MC3T3-E1 cells and reverses the antiproliferative effect of PD 98059; increases the expression of the osteogenic differentiation markers Runx2, Type 1 collagen, and osteocalcin

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6,246

Cayman Chemical A-485, Purity: ≥98% (mixture of isomers), CAS: 1889279-16-6, 10 mg

A p300/CBP inhibitor (IC50 = 60 nM); decreases H3K27Ac levels in PC3 cells; reduces proliferation of various tumor cell lines; inhibits expression of PSA and H3K27Ac occupancy at the PSA enhancer in LNCaP-FGC cells; reduces tumor volume in a LuCaP-77 mouse xenograft model of castration-resistant prostate cancer at 100 mg twice per day for 21 days

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6,247

Cayman Chemical ND-646, Purity: ≥98%, CAS: 1434639-57-2, 5 mg

An ACC inhibitor (IC50s = 3.5 and 4.1 nM for human ACC1 and ACC2, respectively); inhibits production of palmitate and total fatty acid content in A549 cells at 500 nM; induces apoptosis and ER stress in A549 cells at 500 nM; inhibits fatty acid synthesis and reduces tumor growth in an A549 mouse xenograft model at 25 mg/kg twice per day

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6,248

eMolecules 2564-83-2 | TEMPO | Oakwood Chemicals | MFCD00873840 | 157.257 | C9H19NO | 99.000 | CC1(C)CCCC(C)(C)N1O | 1g | 480112099

TEMPO | Oakwood Chemicals | 2564-83-2 | MFCD00873840 | 157.257 | C9H19NO | 99.000 | CC1(C)CCCC(C)(C)N1O | 1g | 480112099

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6,249

Cayman Chemical (–)-Rasfonin, Purity: ≥95%, CAS: 303156-68-5, 5 mg

A fungal metabolite; inhibits concanavalin A- and LPS-induced proliferation of mouse splenocytes (IC50s = 0.7 and 0.5 μg/ml, respectively)

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6,250

Cayman Chemical AA147, Purity: ≥95%, CAS: 393121-74-9, 5 mg

An ER proteostasis regulator; activates an ATF6-dependent ER stress response element reporter and antioxidant response element reporter in HT22 hippocampal cells (EC50s = 3.6 and 3.92 µM, respectively) and protects against glutamate-induced cytotoxicity and prevents increases in ROS in HT22 cells at 10 µM; reduces tunicamycin-induced cell death and increases ERAD in neonatal rat ventricular myocytes at 10 µM; reduces the myocardial, renal, and cerebral infarct size as a percentage of the area at risk in mouse models of ischemia-reperfusion injury induced by LAD ligation, renal portal system occlusion, or MCAO, respectively at 2 mg/kg; prevents the production of NS5 in dengue virus-infected Huh7 cells (IC50 = ~1 µM)

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6,251

Selleck Chemical LLC DT-061 S8774-10MM/1ML

DT-061 (SMAP) is a bioavailable PP2A activator It decreases cell viability in HCC827 and HCC3255 cell lines with IC50 values of 14 3 M and 12 4 M respectively

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6,252

Medchemexpress LLC Metrizoic acid (Metrizoate) | 1949-45-7 | MFCD00867964 | 98.0% | 1 ML

Metrizoic acid (Metrizoate) is an ionic contrast medium. It demonstrates high osmolality and poses a risk of inducing allergic reactions. It is intended for research use only and is not available for sale to patients.

Ionic contrast medium
High osmolality
For research use only
Not for sale to patients

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6,253

Selleck Chemical LLC A-443654-E1125-5MG

A-443654 a derivative of indazole pyridine compounds is a pan Akt (Akt1 2 3 isoforms) inhibitor which binds to the ATP-binding site of Akt It is an ATP competitive and reversible inhibitor

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6,254

Selleck Chemical LLC TR-107 E1986-5MG

TR-107 is a chemical activator of the human mitochondrial protease ClpP with an EC50 of 140 nM It exhibits excellent potency and specificity in the research of triple-negative breast cancer (TNBC) cell models

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6,255

Enzo Life Sciences Neratinib (free base) (10mg). CAS: 698387-09-6

Neratinib is a potent and selective inhibitor of EGFR and HER2. Alternative name: HKI-272. Purity: ≥99% (HPLC). Solubility: Soluble in DMSO at 2 mg/mL. Long Term Storage: -20°C.

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Bioactive Small Molecules

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Medchemexpress LLC Spiroxamine | 118134-30-8 | 99.9% | 50 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Fluralaner (Standard) | 864731-61-3 | 100.0% | 556.29 | 25 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Metrizoic acid (Metrizoate) | 1949-45-7 | MFCD00867964 | 98.0% | 1 ML Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Spiroxamine | 118134-30-8 | 99.9% | 50 MG

Medchemexpress LLC Fluralaner (Standard) | 864731-61-3 | 100.0% | 556.29 | 25 MG

Medchemexpress LLC Metrizoic acid (Metrizoate) | 1949-45-7 | MFCD00867964 | 98.0% | 1 ML